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Popis: A novel, selective inhibitor of receptor-mediated calcium entry. It inhibits receptor-mediated calcium entry in stimulated platelets (IC50=8-12µM) neutrophils and endothelial cells at concentrations which do not affect internal Ca²⁺ release. Note, in some cells SK&F 96365 can activate a novel Ca²⁺ entry pathway. Blocks TRPC3 and TRPC6 activation. Inhibits the histamine-induced formation of nitric oxide in human endothelial cells.
Katalogové číslo: ENZOBMLCA2300025
Měrná jednotka: 1 * 25 mg
Dodavatel: ENZO LIFE SCIENCES


Popis: SKF-96365 hydrochloride ≥99%
Katalogové číslo: J60937.MF
Měrná jednotka: 1 * 50 mg
Dodavatel: Thermo Fisher Scientific

Popis: Proadifen hydrochloride 95%
Katalogové číslo: ACRO457880050
Měrná jednotka: 1 * 5 g
Dodavatel: Thermo Fisher Scientific


Popis: Cytochrome P450 inhibitor
Katalogové číslo: ENZOBMLEI1051000
Měrná jednotka: 1 * 1 g
Dodavatel: ENZO LIFE SCIENCES


Popis: Potent antitumor agent. Inhibitor of DNA-topoisomerase. Analog of (S)-(⁺)-camptothecin. Used in chemotherapy of several different cancers.
Katalogové číslo: ENZOALX350133M025
Měrná jednotka: 1 * 25 mg
Dodavatel: ENZO LIFE SCIENCES


Popis: Proadifen hydrochloride
Katalogové číslo: J63833.03
Měrná jednotka: 1 * 1 g
Dodavatel: Thermo Fisher Scientific

Popis: Topotecan hydrochloride hydrate 97%
Katalogové číslo: 467182500.
Měrná jednotka: 1 * 250 mg
Dodavatel: Thermo Fisher Scientific

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Popis: MAPK/ERK Signalling Pathway
Katalogové číslo: APOSBISN0228-10MG
Měrná jednotka: 1 * 10 mg
Dodavatel: Apollo Scientific


Popis: A potent irreversible inactivator of calmodulin. Possesses potent antiproliferative and cytotoxic activity. It is also an irreversible D2 dopamine receptor antagonist.
Katalogové číslo: ENZOBMLCA3250050
Měrná jednotka: 1 * 50 mg
Dodavatel: ENZO LIFE SCIENCES


Popis: Demethylase inhibitor
Katalogové číslo: ENZOBMLEI2170001
Měrná jednotka: 1 * 1 g
Dodavatel: ENZO LIFE SCIENCES


Popis: Phosphodiesterase 9A is a cGMP-specific phosphodiesterase. PDE9A activity is inhibited by zaprinast, but it is insensitive to rolipram, vinpocetine, SKF-94120, dipyridamole, and IBMX. More than 20 alternatively spliced variants have been reported (Rentero et al. 2003). PDE9A has been implicated in penile erectile dysfunction, as well as in functional disturbances in which intraneuronal signal transmission via second messengers are important in the pathophysiology (example, bipolar affective disorder). PDE9A is the only cGMP-specific PDE with significant expression in the forebrain, and as such is likely to function in NO-cGMP signaling.
Katalogové číslo: PRSI48-318
Měrná jednotka: 1 * 50 µG
Dodavatel: ProSci Inc.


Popis: SKF-96365 HYDROCHLORIDE 1 * 1 mg
Katalogové číslo: CAYM10009312-1
Měrná jednotka: 1 * 1 mg
Dodavatel: Cayman Chemical


Popis: L(+)-cystein hydrochlorid monohydrát, TECHNICAL
Katalogové číslo: 23255.186
Měrná jednotka: 1 * 100 g
Dodavatel: VWR Chemicals

Popis: SKF-96365 HYDROCHLORIDE 1 * 50 mg
Katalogové číslo: CAYM10009312-50
Měrná jednotka: 1 * 50 mg
Dodavatel: Cayman Chemical


Popis: SKF-96365 HYDROCHLORIDE 1 * 10 mg
Katalogové číslo: CAYM10009312-10
Měrná jednotka: 1 * 10 mg
Dodavatel: Cayman Chemical


Popis: L(+)-Ornithine hydrochloride ≥99%
Katalogové číslo: 0958-500G
Měrná jednotka: 1 * 500 g
Dodavatel: VWR Chemicals

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